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EPZ020411 2HCl
CAS No. ——
EPZ020411 2HCl ( —— )
Catalog No. M17704 CAS No. ——
EPZ020411 is an effective and specific small molecule PRMT6 inhibitor (IC50=10 nM).
Purity : >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| Size | Price / USD | Stock | Quantity |
| 5MG | 189 | Get Quote |
|
| 10MG | 301 | Get Quote |
|
| 25MG | 627 | Get Quote |
|
| 100MG | Get Quote | Get Quote |
|
| 200MG | Get Quote | Get Quote |
|
| 500MG | Get Quote | Get Quote |
|
| 1G | Get Quote | Get Quote |
|
Biological Information
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Product NameEPZ020411 2HCl
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NoteResearch use only, not for human use.
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Brief DescriptionEPZ020411 is an effective and specific small molecule PRMT6 inhibitor (IC50=10 nM).
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DescriptionEPZ020411 is an effective and specific small molecule PRMT6 inhibitor (IC50=10 nM).
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In Vitro——
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In Vivo——
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Synonyms——
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PathwayImmunology/Inflammation
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TargetTLR
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RecptorPRMT6|PRMT1|PRMT8
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Research Area——
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Indication——
Chemical Information
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CAS Number——
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Formula Weight515.51
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Molecular FormulaC25H40Cl2N4O3
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Purity>98% (HPLC)
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Solubility——
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SMILESCl.Cl.CNCCN(C)Cc1cnnc1c2ccc(cc2)O[C@H]4C[C@H](OCCC3CCOCC3)C4
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Chemical Name——
Shipping & Storage Information
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Storage(-20℃)
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ShippingWith Ice Pack
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Stability≥ 2 years
Reference
1.Mitchell LH, et al. Aryl Pyrazoles as Potent Inhibitors of Arginine Methyltransferases: Identification of the First PRMT6 ToolCompound. ACS Med Chem Lett. 2015 Apr 6;6(6):655-659.
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